August 21, 2.30 pm in AG-80
Title :
Molecular Knots and Antimicrobial Peptides
Abstract :
Molecules with complex topologies, such as molecular links and knots, are often found in nature, but remain extremely difficult to synthesize using the current methods of chemistry. Over the past 30 years, the only strategy for the synthesis of molecular knots has been reliant on metal templation.1 Through our work on dynamic disulfide chemistry, we established that the hydrophobic effect can provide a powerful alternative synthetic strategy that enabled us to synthesize a variety of different knots, some of which had remained elusive until now: Hopf links,2,3 Solomon links,4 trefoil knots,5 and figure eight knots.4 In some cases, the hydrophobic effect overcomes electrostatic interactions between electron-rich and electron-deficient aromatic units, leading to the formation of unconventional structures that seem to contradict the current models of donor-acceptor interactions. A mechanism that succeeds in rationalizing and predicting their formation was proposed. This mechanism represents a major advance in understanding the role of hydrophobic effect in the assembly of complex architectures
In the second part of my talk, I will outline my current work on human defensins 5 and 6 (HD5-6), small (2-5 kDa) cysteine-rich host-defense peptides, which are key contributors to innate immunity and provides the first line of defense for detection and response to microbial invasion.6 Paneth cells protect the intestinal epithelium against infection and colonization of pathogenic or opportunistic microbes by secreting a mixture of antimicrobial peptides and proteins that includes HD5 and HD6. Although both peptides exhibit a common tertiary structure, they possess unique functional attributes. HD5 has broad-spectrum antibacterial activity in vitro. In contrast, HD6 provides only negligible antimicrobial activity in vitro but forms nanonets-like higher-order oligomeric structures that entrap bacteria in the intestinal lumen in order to prevent invasion. In the oxidized forms, both defensins contain three conserved and regiospecific intramolecular disulfide bonds. We explored the redox properties of these disulfide bonds and their role to maintain the peptides antimicrobial function. These peptides can interact with various metals, notably zinc,7 an important metal controlling the immune response.
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- March 24, 2014 at 4.00 pm in AG-69
- March 20, 2014 at 2.30 pm in AG-80
- March 10, 2014 at 4.00 pm in AG-69
- March 3, 2014 at 4.00 pm in AG-69
- February 25, 2014 at 2.30 pm in B-333 (DBS Seminar Room)
- February 19, 2014 at 2.30 pm in AG-69
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- February 17, 2014 at 4.00 pm in AG-69
- February 12, 2014 at 2.30 pm in D-406
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- January 30, 2014 at 11.30 am in NMR Seminar Room
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- October 29, 2013 at 11.30 am in AG-80
- October 28, 2013 at 4.00 pm in AG-69
- October 22, 2013 at 11.30 am in AG-80
- October 21, 2013 at 4.00 pm in AG-69
- October 15, 2013 at 11.30 am in AG-80
- October 14, 2013 at 4.00 pm in AG-69
- September 26th & 27th, 2013 in AG-66
- September 23, 4.00 pm in AG-69
- August 19, 2013 at 4.00 pm in AG69
- August 5, 2013 at 4.00 pm in AG69
- July 1, 2013 at 4.00 pm in AG69
- June 17, 2013 at 4.00 pm in AG69
- June 10, 2013 at 4.00 pm in AG69
- May 27, 2013 at 4.00 pm in AG69
- May 6, 2013 at 4.00 pm in AG66
- May 9, 2013 at 2.30 pm in AG80
- April 29, 2013 at 4.00 pm in AG69
- April 22, 2013 at 4.00 pm in AG69
- April 18, 2013 at 2.30 pm in AG80
- April 12, 2013 at 2.30 pm in AG80
- April 15, 2013 at 4.00 pm in AG69
- April 11, 2013 at 2.30 pm in AG80
- April 10, 2013 at 11.30 am in NMR Conference Room
- April 8, 2013 at 4.00 pm in AG69
- April 5, 2013 at 2.30 pm in AG69
- April 3, 2013 at 2.30 pm in AG69
- March 28, 2013 at 4.00 pm in AG80
- March 25, 2013 at 4.00 pm in AG69
- March 22, 2013 at 2.30 pm in AG80
- March 21, 2013 at 2.30 pm in AG80
- March 18, 2013 at 4.00 pm in AG69
- March 14, 2013 at 2.30 pm in AG80
- March 11, 2013 at 4.00 pm in AG69
- March 6, 2013 at 2.30 pm in NMR Conference Room
- March 5, 2013 at 2.30 pm in DBS Seminar Room (B-333)
- March 4, 2013 at 4.00 pm in AG66
- February 27, 2013 at 11.30 am in AG66
- February 25, 2013 at 2.30 pm in AG69
- February 18, 2013 at 4.00 pm in AG69
- February 15, 2013 at 2.30 pm in AG80
- February 14, 2013 at 2.30 pm in AG80
- January 30, 2013 at 11.30 am in AG80
- January 29, 2013 at 4.00 pm in AG80
- January 28, 2013 at 4.00 pm in AG69
- January 23, 2013 at 11.30 am in AG69
- January 21, 2013 at 4.00 pm in AG69
- January 17, 2013 at 2.30 pm in AG80
- January 14, 2013 at 4.00 pm in AG69
- January 7, 2013 at 4.00 pm in AG80
- May 20, 2013 at 4.00 pm in AG69
- June 3, 2013 at 4.00 pm in AG69